• Tranexamic Acid

Tranexamic Acid

The Synthetic Whitening Derivative for Quick and Safe Brightening

Tranexamic Acid is a synthetic derivative of aminomethylbenzoic acid, known for its Anti-fibrinolytic activity. It has a strong affinity for the five lysine binding sites of plasminogen. It is highly valued for its efficacy in making skin white and bright quickly (within 1-2 weeks) with quick effect products.

CAS No.

1197-18-8

Appearance Color

White Powder

Key Efficacy

Anti-Chloasma (Melasma), Whitening, Anti-Fibrinolytic, Spot Reduction

Solubility

Soluble in water

Stability

High thermal stability, good stability, not easily discolored

Break the Formulation Bottleneck: The Clinically Superior, High-Stability Whitening Alternative for Next-Gen Clean Beauty

Are your formulators struggling with the instability, skin irritation, and complex handling of traditional spot-fading actives like Hydroquinone? In today’s highly competitive skincare market, consumers demand rapid results without compromising skin barrier health. Elevate your brand with our premium Tranexamic Acid—a highly stable, exceptionally compatible, and clinically validated active ingredient designed to deliver rapid brightening with a superior safety profile.

1. Clinical Data First: Proven Efficacy Meets Uncompromising Safety

We back our active ingredients with rigorous clinical data, providing you with the authoritative proof needed to build consumer trust. In a 12-week clinical study comparing a 3% Tranexamic Acid solution against the industry gold standard (3% Hydroquinone + 0.01% Dexamethasone) for treating chloasma/melasma:

  • Unmatched Safety: The Tranexamic Acid group reported a mere 20% side effect rate, drastically outperforming the Hydroquinone combination group which suffered a 48% side effect rate.

  • Equivalent Efficacy: Tranexamic Acid demonstrated a comparable cumulative effect in reducing the Melasma Area and Severity Index (MASI) score, dropping from 31.68 at baseline down to 12.01.

  • Rapid Results: Clinical feedback confirms visible skin brightening and whitening effects within just 1 to 2 weeks of use.

2. Strategic Business Value

For High-End Beauty Brands: The Ultimate “Clean Beauty” Choice

Consumers are actively rejecting harsh chemicals. Tranexamic Acid offers the perfect marketing narrative: a highly effective, dermatologist-backed active that acts powerfully against hyperpigmentation but is remarkably gentle on the skin. It possesses a significantly lower toxicity profile than aminocaproic acid, making it the premier choice for premium, clean-label brightening serums, anti-chloasma treatments, and spot corrector fluids.

For Senior Formulators: Ultimate Formula Compatibility

Say goodbye to the thermal instability and discoloration issues common with traditional Vitamin C derivatives or Hydroquinone. Our Tranexamic Acid is characterized by extremely low irritation (safe even for extended-wear facial masks) and unmatched versatility. It is highly resistant to heat, does not easily discolor over time, and integrates seamlessly into complex cosmetic chassis.

3. Core Product Specifications

Parameter Specification
INCI Name Tranexamic Acid
CAS Number 1197-18-8
Appearance Colorless, odorless powder
Solubility Easily soluble in water
Purity ≥ 95.0%
Heavy Metals < 10ppm
Recommended Dosage 0.1% – 1.0%

4. Precision Mechanism of Action (MoA)

Tranexamic Acid operates at the root of melanogenesis by intercepting the inflammatory pathways that trigger pigment production:

  • Plasmin Inhibition: It effectively blocks the conversion of plasminogen into plasmin.

  • Melanogenesis Blockade: It disrupts the UV-induced keratinocyte PA system, effectively preventing the formation of melanin—a crucial factor in preventing and treating chloasma.

  • Inflammatory Factor Reduction: It suppresses the release of inflammatory and injury factors (triggered by UV light or skin trauma) that typically stimulate melanocytes via the Plasmin/FGF pathway.

5. Ready-to-Use Solutions: Golden Formula Inspirations

Accelerate your R&D process with our highly recommended, synergistic active combinations designed for maximum efficacy:

  • The Complete Melanin Blocker (Tranexamic Acid + Niacinamide): A dual-action powerhouse. Tranexamic Acid inhibits melanin synthesis at the source via anti-plasmin action, while Niacinamide prevents the transfer of existing melanin to the epidermis.

  • The Antioxidant Radiance Booster (Tranexamic Acid + Vitamin C): Combines targeted spot-prevention with broad-spectrum antioxidant protection, maximizing overall skin radiance and tone uniformity.

6. Quality Assurance & Factory Certifications

We are committed to the highest global standards of purity, safety, and regulatory compliance. Our production facilities and quality management systems are backed by:

  • COSMOS (Natural and Organic Cosmetic Standard)

  • ISO 9001

  • ISO 22000

  • HALAL Certification

  • IQNET (The International Certification Network)

Source the Clinically Superior Tranexamic Acid for Safe, Fast, and Effective Whitening Formulations.

🔒 Get Your Technical Dossier: Contact us now to access the full TDS, MSDS, COA, and detailed Clinical Efficacy Reports.

🔬 Apply for a Free Sample: Experience the high solubility, exceptional stability, and low-irritation profile in your own lab today.

📞 Get a Customized Quote: Reach out to our B2B technical sales team to discuss bulk pricing, lead times, and high-purity specifications tailored to your brand’s needs.

Natural huataiは、高純度のグラブリジン(美白)、リコカルコンA(抗ニキビ)、トタロール、グリチルリチン酸ジカリウムを特徴とする、先進的な機能性スキンケア原料を専門としています。当社は、オーダーメイドの濃度(1%–99%)と包括的なOEMソリューションを提供しています。ISO 9001/22000およびCOSMOS認証を取得した当社の生産施設は、世界のビューティーブランドにプレミアムな化粧品グレードの品質を保証します。

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